BX-912 [Ligand Id: 8007] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| 3-phosphoinositide dependent protein kinase 1 in Human [GtoPdb: 1519] [UniProtKB: O15530] | ||||||||
| GtoPdb | In a direct kinase activity measuring phosphorylation od a small peptide substrate mimetic | - | 7.59 | pIC50 | 26 | nM | IC50 | J Biol Chem (2005) 280: 19867-74 [PMID:15772071] |
| protein kinase A in Human [GtoPdb: 1694] | ||||||||
| GtoPdb | - | - | 6.96 | pIC50 | 110 | nM | IC50 | J Biol Chem (2005) 280: 19867-74 [PMID:15772071] |
| kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968] | ||||||||
| GtoPdb | - | - | 6.39 | pIC50 | 410 | nM | IC50 | J Biol Chem (2005) 280: 19867-74 [PMID:15772071] |
| cyclin dependent kinase 2 in Human [GtoPdb: 1973] [UniProtKB: P24941] | ||||||||
| GtoPdb | - | - | 6.19 | pIC50 | 650 | nM | IC50 | J Biol Chem (2005) 280: 19867-74 [PMID:15772071] |
| checkpoint kinase 1 in Human [GtoPdb: 1987] [UniProtKB: O14757] | ||||||||
| GtoPdb | - | - | 6.08 | pIC50 | 830 | nM | IC50 | J Biol Chem (2005) 280: 19867-74 [PMID:15772071] |
| glycogen synthase kinase 3 beta in Human [GtoPdb: 2030] [UniProtKB: P49841] | ||||||||
| GtoPdb | - | - | 5.13 | pIC50 | 7400 | nM | IC50 | J Biol Chem (2005) 280: 19867-74 [PMID:15772071] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
