I-BRD9 [Ligand Id: 8397] activity data from GtoPdb

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  • bromodomain containing 9 in Human [GtoPdb: 2728] [UniProtKB: Q9H8M2]
  • This target only has 0 pki data point
1 _lig_chart_1 bromodomain containing 9 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
bromodomain containing 9 in Human [GtoPdb: 2728] [UniProtKB: Q9H8M2]
GtoPdb Binding affinity for endogenous BRD9 from HuT-78 cell lysates, measured in a chemoproteomic competition binding assay followed by Western blot analysis. - 7.1 pIC50 79.4 nM IC50 J. Med. Chem. (2016) 59: 1425-39 [PMID:25856009]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.