S-BMPA [Ligand Id: 8676] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL90403 |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Carboxypeptidase A3 (mast cell)/Mast cell carboxypeptidase A in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2645] [GtoPdb: 1589] [UniProtKB: P15088] | ||||||||
| ChEMBL | Compound was tested for inhibitory activity against carboxypeptidase A | B | 8.11 | pKi | 7.8 | nM | Ki | Bioorg Med Chem Lett (1993) 3: 2681-2684 |
| Carboxypeptidase A1 (pancreatic) in Bovine [GtoPdb: 1587] | ||||||||
| GtoPdb | - | - | 8.11 | pKi | 7.8 | nM | Ki | Bioorg Med Chem Lett (1993) 3: 2681-2684 |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
