compound 13b [PMID: 19101153] [Ligand Id: 8808] activity data from GtoPdb and ChEMBL

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

ChEMBL ligand: CHEMBL473744
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
ABCC9/Sulfonylurea receptor 2 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1971] [GtoPdb: 2746] [UniProtKB: O60706]
GtoPdb - - 6.17 pEC50 670 nM EC50 Bioorg. Med. Chem. (2009) 17: 855-66 [PMID:19101153]
ChEMBL Channel opening activity at SUR2B/Kir6.2 potassium ATP channel in human TE671 cells assessed as isometric force by FLIPR B 6.17 pEC50 670 nM EC50 Bioorg. Med. Chem. (2009) 17: 855-866 [PMID:19101153]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]