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ChEMBL ligand: CHEMBL3183531 |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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lysine demethylase 5B in Human [GtoPdb: 2681] [UniProtKB: Q9UGL1] | ||||||||
GtoPdb | - | - | 5.01 | pIC50 | 9700 | nM | IC50 | Nature (2014) 514: E1-2 [PMID:25279926] |
lysine demethylase 5C in Human [GtoPdb: 2682] [UniProtKB: P41229] | ||||||||
GtoPdb | - | - | 4.82 | pIC50 | 15000 | nM | IC50 | Nature (2014) 514: E1-2 [PMID:25279926] |
lysine demethylase 6A in Human [GtoPdb: 2684] [UniProtKB: O15550] | ||||||||
GtoPdb | - | - | 5.18 | pIC50 | 6600 | nM | IC50 | Nature (2014) 514: E1-2 [PMID:25279926] |
lysine demethylase 6B in Human [GtoPdb: 2685] [UniProtKB: O15054] | ||||||||
GtoPdb | - | - | 5.07 | pIC50 | 8600 | nM | IC50 | Nature (2014) 514: E1-2 [PMID:25279926] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]