erdafitinib [Ligand Id: 9039] activity data from GtoPdb

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  • fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362]
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  • fibroblast growth factor receptor 2 in Human [GtoPdb: 1809] [UniProtKB: P21802]
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  • fibroblast growth factor receptor 3 in Human [GtoPdb: 1810] [UniProtKB: P22607]
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  • fibroblast growth factor receptor 4 in Human [GtoPdb: 1811] [UniProtKB: P22455]
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  • kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362]
GtoPdb - - 8.94 pIC50 1.14 nM IC50 WO2011135376 A1. Pyrazolyl quinazoline kinase inhibitors. (2011)
fibroblast growth factor receptor 2 in Human [GtoPdb: 1809] [UniProtKB: P21802]
GtoPdb - - 8.64 pIC50 2.29 nM IC50 WO2011135376 A1. Pyrazolyl quinazoline kinase inhibitors. (2011)
fibroblast growth factor receptor 3 in Human [GtoPdb: 1810] [UniProtKB: P22607]
GtoPdb - - 8.52 pIC50 3.02 nM IC50 WO2011135376 A1. Pyrazolyl quinazoline kinase inhibitors. (2011)
fibroblast growth factor receptor 4 in Human [GtoPdb: 1811] [UniProtKB: P22455]
GtoPdb - - 8.25 pIC50 5.62 nM IC50 WO2011135376 A1. Pyrazolyl quinazoline kinase inhibitors. (2011)
kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968]
GtoPdb - - 7.44 pIC50 36.3 nM IC50 WO2011135376 A1. Pyrazolyl quinazoline kinase inhibitors. (2011)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.