PZM21 [Ligand Id: 9286] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372]
GtoPdb - - 8.96 pKi 1.1 nM Ki Nature (2016) 537: 185-190 [PMID:27533032]
GtoPdb In a Gi/o activation assay. - 8.34 pEC50 4.6 nM EC50 Nature (2016) 537: 185-190 [PMID:27533032]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.