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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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mechanistic target of rapamycin kinase in Human [GtoPdb: 2109] [UniProtKB: P42345] | ||||||||
GtoPdb | In a biochemical assys using recombinant wild type enzyme. | - | 7.82 | pIC50 | 15 | nM | IC50 | Medchemcomm (2016) 7: 471-477 |
GtoPdb | In a cell viability assay. | - | 8.05 | pEC50 | 9 | nM | EC50 | Medchemcomm (2016) 7: 471-477 |
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336] | ||||||||
GtoPdb | In a biochemical assay. | - | 6.01 | pIC50 | 981 | nM | IC50 | Medchemcomm (2016) 7: 471-477 |
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329] | ||||||||
GtoPdb | In a biochemical assay. | - | 5.74 | pIC50 | 1840 | nM | IC50 | Medchemcomm (2016) 7: 471-477 |
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736] | ||||||||
GtoPdb | In a biochemical assay. | - | 5.87 | pIC50 | 1340 | nM | IC50 | Medchemcomm (2016) 7: 471-477 |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.