compound 46c [PMID: 29350534] [Ligand Id: 9883] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CXCR4 in Human [GtoPdb: 71] [UniProtKB: P61073] | ||||||||
| GtoPdb | Measuring antagonist-mediated inhibition of CXCL12-induced calcium flux in human T lymphoblast CCRF-CEM cells. | - | 7.81 | pIC50 | 15.5 | nM | IC50 | J Med Chem (2018) 61: 946-979 [PMID:29350534] |
| CXCR4 in Mouse [GtoPdb: 71] [UniProtKB: P70658] | ||||||||
| GtoPdb | - | - | 8.03 | pIC50 | 9.24 | nM | IC50 | J Med Chem (2018) 61: 946-979 [PMID:29350534] |
| CYP2D6 in Human [GtoPdb: 1329] [UniProtKB: P10635] | ||||||||
| GtoPdb | - | - | 5.58 | pIC50 | 2610 | nM | IC50 | J Med Chem (2018) 61: 946-979 [PMID:29350534] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
