Synonyms: BAL-9141 | BAL9141 | BAL9141-000 | BAL9141000 | Ro-63-9141 | Ro-639141 | Zeftera® | Zevtera®
ceftobiprole is an approved drug (UK (2013), FDA (2024))
Compound class:
Synthetic organic
Comment: Ceftobiprole is a clinical stage, broad-spectrum, fifth-generation, pyrrolidinone cephalosporin antibacterial [3]. It was developed as a treatment for hospital-acquired pneumonia (HAP) and community-acquired pneumonia (CAP), in particular those infections caused by methicillin-resistant Staphylococcus aureus (MRSA). In clinical trials ceftobiprole is administered by intravenous infusion as the water-soluble prodrug ceftobiprole medocaril (BAL5788; PubChem CID 135413544).
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Classification ![]() |
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Compound class | Synthetic organic |
Approved drug? | Yes (UK (2013), FDA (2024)) |
Approved drug? | Yes. UK (2013) |
International Nonproprietary Names ![]() |
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INN number | INN |
8531 | ceftobiprole |
Synonyms ![]() |
BAL-9141 | BAL9141 | BAL9141-000 | BAL9141000 | Ro-63-9141 | Ro-639141 | Zeftera® | Zevtera® |
Database Links ![]() |
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Specialist databases | |
Antibiotic DB
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Ceftobiprole (active moiety of ceftobiprole medocaril) |
Other databases | |
CAS Registry No. | 209467-52-7 (source: WHO INN record) |
ChEMBL Ligand | CHEMBL520642 |
GtoPdb PubChem SID | 405560228 |
PubChem CID | 135413542 |
Search Google for chemical match using the InChIKey | VOAZJEPQLGBXGO-SDAWRPRTSA-N |
Search Google for chemicals with the same backbone | VOAZJEPQLGBXGO |
Search PubMed clinical trials | ceftobiprole |
Search PubMed titles | ceftobiprole |
Search PubMed titles/abstracts | ceftobiprole |
UniChem Compound Search for chemical match using the InChIKey | VOAZJEPQLGBXGO-SDAWRPRTSA-N |
UniChem Connectivity Search for chemical match using the InChIKey | VOAZJEPQLGBXGO-SDAWRPRTSA-N |
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Ceftobiprole (links to external site)
Cat. No. HY-112579 |