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Synonyms: OBE101 [2] | SERC® | Vasomotal®
betahistine is an approved drug (FDA (1970s))
Compound class:
Synthetic organic
Comment: This is an orally delivered histamine receptor modulator that has weak agonist activity at histamine H1 receptors and more potent antagonist activity at the H3 receptor subtype [1].
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Classification ![]() |
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Compound class | Synthetic organic |
Approved drug? | Yes. US FDA (1970) |
Withdrawn drug? | Yes |
International Nonproprietary Names ![]() |
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INN number | INN |
1502 | betahistine |
Synonyms ![]() |
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OBE101 [2] | SERC® | Vasomotal® |
Database Links ![]() |
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CAS Registry No. | 5638-76-6 (source: PubChem) |
ChEMBL Ligand | CHEMBL24441 |
DrugBank Ligand | DB06698 |
GtoPdb PubChem SID | 461663492 |
PubChem CID | 2366 |
Search Google for chemical match using the InChIKey | UUQMNUMQCIQDMZ-UHFFFAOYSA-N |
Search Google for chemicals with the same backbone | UUQMNUMQCIQDMZ |
Search PubMed clinical trials | betahistine |
Search PubMed titles | betahistine |
Search PubMed titles/abstracts | betahistine |
UniChem Compound Search for chemical match using the InChIKey | UUQMNUMQCIQDMZ-UHFFFAOYSA-N |
UniChem Connectivity Search for chemical match using the InChIKey | UUQMNUMQCIQDMZ-UHFFFAOYSA-N |
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Betahistine (links to external site)
Cat. No. HY-B0524 |