Synonyms: MMV687696 | Q203
Compound class:
Synthetic organic
Comment: Telacebec is a first-in-class imidazopyridine amide that inhibits the mycobacterial cytochrome bc1 complex [3]. It is being clinically evaluated as a treatment for tuberculosis (TB).
Telacebec was one of the compounds with activity against Mycobacterium tuberculosis included in the Medicines for Malaria Venture (MMV) Pathogen Box (see MMVOpen for futher details). |
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Classification | |
Compound class | Synthetic organic |
IUPAC Name |
6-chloro-2-ethyl-N-[[4-[4-[4-(trifluoromethoxy)phenyl]piperidin-1-yl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide |
International Nonproprietary Names | |
INN number | INN |
10573 | telacebec |
Synonyms |
MMV687696 | Q203 |
Database Links | |
Specialist databases | |
Antibiotic DB | Q203, Telacebec |
Other databases | |
BindingDB Ligand | 50022086 |
CAS Registry No. | 1334719-95-7 (source: Scifinder) |
ChEMBL Ligand | CHEMBL3298910 |
DrugBank Ligand | DB17754 |
GtoPdb PubChem SID | 485206074 |
PubChem CID | 68234908 |
RCSB PDB Ligand | HUU |
Search Google for chemical match using the InChIKey | OJICYBSWSZGRFB-UHFFFAOYSA-N |
Search Google for chemicals with the same backbone | OJICYBSWSZGRFB |
Search PubMed clinical trials | telacebec |
Search PubMed titles | telacebec |
Search PubMed titles/abstracts | telacebec |
UniChem Compound Search for chemical match using the InChIKey | OJICYBSWSZGRFB-UHFFFAOYSA-N |
UniChem Connectivity Search for chemical match using the InChIKey | OJICYBSWSZGRFB-UHFFFAOYSA-N |