Synonyms: LY-3819469 | LY3819469
Compound class:
Nucleic acid
Comment: Lepodisiran (LY3819469) is an apolipoprotein A synthesis reducer. It is a GalNac-conjugated short interfering RNA (siRNA) that was designed to treat atherosclerotic cardiovascular disease in patients with elevated lipoprotein A [1-2].
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Classification ![]() |
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Compound class | Nucleic acid |
Compound subclass | siRNA |
Target | apolipoprotein A |
International Nonproprietary Names ![]() |
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INN number | INN |
13068 | lepodisiran |
Synonyms ![]() |
LY-3819469 | LY3819469 |
Database Links ![]() |
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CAS Registry No. | 2808361-18-2 (source: WHO INN record) |
GtoPdb PubChem SID | 507750342 |
Search PubMed clinical trials | lepodisiran |
Search PubMed titles | lepodisiran |
Search PubMed titles/abstracts | lepodisiran |