t-Boc-FLFLF   Click here for help

GtoPdb Ligand ID: 1030

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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
FPR1 Hs Antagonist Antagonist 6.0 – 6.5 pKi - 5
pKi 6.0 – 6.5 [5]
FPR1 Hs Antagonist Antagonist 6.6 pIC50 - 4
pIC50 6.6 [4]
FPR2/ALX Hs Antagonist Antagonist 4.3 – 6.0 pIC50 - 1-3
pIC50 4.3 – 6.0 [1-3]