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Synonyms: 125I-Sarcosine1, D-Alanine8-Angiotensin II
Compound class:
Peptide or derivative
Comment: This is a radiolabelled version of the angiotensin II analogue Sarcosine1, D-Alanine8-Ang II (TRV027) that was developed by Trevena. TRV027 is β-arrestin biased agonist of angiotensin receptor activation.
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| Bioactivity Comments |
| This is a low potency AT1 receptor agonist [1], likely due to the D-Ala substitution at position 8. |
