BIM 23027   Click here for help

GtoPdb Ligand ID: 2033

Synonyms: BIM23027
Comment: Cyclic peptide
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST2 receptor Mm Agonist Full agonist 10.2 – 12.0 pIC50 - 3-4
pIC50 10.2 – 12.0 [3-4]
SST2 receptor Hs Agonist Agonist 10.9 pIC50 - 1
pIC50 10.9 (IC50 1.4x10-11 M) [1]
SST2 receptor Rn Agonist Agonist 9.7 pIC50 - 2
pIC50 9.7 (IC50 2x10-10 M) [2]