R-486   Click here for help

GtoPdb Ligand ID: 2105

Synonyms: [Trp7,β-Ala8]neurokinin A(4-10) | MEN 10295 | R 486 | R486
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
NK1 receptor Hs Antagonist Antagonist 6.5 – 6.6 pKi - 1
pKi 6.5 – 6.6 [1]