d[Leu4,Dap8]VP   Click here for help

GtoPdb Ligand ID: 2189

Synonyms: [deamino-Cys1,Leu4,Dap8]vasopressin
Comment: Synthetic analogue of AVP
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
V1B receptor Rn Agonist Full agonist 9.4 pKi - 1
pKi 9.4 [1]
OT receptor Rn Agonist Full agonist 6.9 pKi - 1
pKi 6.9 [1]
V2 receptor Rn Agonist Full agonist 6.6 pKi - 1
pKi 6.6 [1]
V1A receptor Rn Agonist Full agonist 5.5 pKi - 1
pKi 5.5 [1]