[D-Pro4,D-Trp7,9,10]substance P (4-11)   

GtoPdb Ligand ID: 6185

Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
BB2 receptor Rn Antagonist Antagonist <5.0 pKi - 2
pKi <5.0 (Ki >1x10-5 M) [2]
BB2 receptor Hs Antagonist Antagonist 5.0 – 5.4 pIC50 - 1
pIC50 5.0 – 5.4 (IC50 1x10-5 – 3.8x10-6 M) [1]