B-9430   Click here for help

GtoPdb Ligand ID: 653

Synonyms: B 9430 | B9430 | D-Arg-[Hyp3,Igl5,D-Igl7,Oic8]-bradykinin
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
B2 receptor Hs Antagonist Antagonist 8.4 pA2 - 2
pA2 8.4 [2]
Description: Apparent affinity for bradykinin B2 receptor in human umbilical vein
B1 receptor Hs Antagonist Antagonist 7.7 pA2 - 2
pA2 7.7 [2]
B1 receptor Mm Antagonist Antagonist 6.1 pA2 - 2
pA2 6.1 [2]
B2 receptor Hs Antagonist Antagonist 8.6 – 9.6 pKi - 1,3
pKi 8.6 – 9.6 [1,3]
B2 receptor Mm Antagonist Antagonist 8.5 – 9.5 pKi - 1
pKi 8.5 – 9.5 [1]
B1 receptor Hs Antagonist Antagonist 7.9 pKi - 1,3
pKi 7.9 [1,3]
B1 receptor Mm Antagonist Antagonist 6.6 pKi - 1
pKi 6.6 [1]