Ligand id: 9221

Name: azapro-3

View interactive charts of activity data from GtoPdb and ChEMBL (where available) across species

Bioactivity Comments
Azapro-3, inhibits free PR3 in solution, PR3 bound to neutrophil membranes, and PR3 in crude lung secretions from patients with chronic inflammatory pulmonary diseases [1].
Selectivity at enzymes
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
proteinase 3 Hs Inhibitor Inhibition 5.8 pKi - 1
pKi 5.8 (Ki 1.5x10-6 M) [1]