P32 [PMID: 27108698]   Click here for help

GtoPdb Ligand ID: 9384

Compound class: Peptide
Comment: Selective C5a2 receptor agonist
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
C5a2 receptor Hs Agonist Biased agonist 3.7 pKi - 1
pKi 3.7 (Ki 2.23x10-4 M) Exhibits selective partial agonism for recruitment of β-arrestin 2 via C5aR2 in a BRET C5aR2-β-arrestin 2 recruitment assay [1]
Description: Binding assay