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Compound class: Peptide or derivative
Ligand Activity Visualisation Charts
These are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts.✖
1. Harland SP, Kuc RE, Pickard JD, Davenport AP. (1995)
Characterization of endothelin receptors in human brain cortex, gliomas, and meningiomas.
J Cardiovasc Pharmacol, 26 Suppl 3: S408-11. [PMID:8587429]
2. Molenaar P, Kuc RE, Davenport AP. (1992)
Characterization of two new ETB selective radioligands, [125I]-BQ3020 and [125I]-[Ala1,3,11,15]ET-1 in human heart.
Br J Pharmacol, 107 (3): 637-9. [PMID:1472961]
3. Peter MG, Davenport AP. (1995)
Selectivity of [125I]-PD151242 for human, rat and porcine endothelin ETA receptors in the heart.
Br J Pharmacol, 114 (2): 297-302. [PMID:7881728]