[Leu8,des-Arg9]bradykinin

Ligand id: 641

Name: [Leu8,des-Arg9]bradykinin

Structure and Physico-chemical Properties

2D Structure
References
1. Aramori I, Zenkoh J, Morikawa N, O'Donnell N, Asano M, Nakamura K, Iwami M, Kojo H, Notsu Y. (1997)
Novel subtype-selective nonpeptide bradykinin receptor antagonists FR167344 and FR173657.
Mol. Pharmacol., 51 (2): 171-6. [PMID:9203620]
2. Austin CE, Faussner A, Robinson HE, Chakravarty S, Kyle DJ, Bathon JM, Proud D. (1997)
Stable expression of the human kinin B1 receptor in Chinese hamster ovary cells. Characterization of ligand binding and effector pathways.
J. Biol. Chem., 272 (17): 11420-5. [PMID:9111052]
3. Bastian S, Loillier B, Paquet JL, Pruneau D. (1997)
Stable expression of human kinin B1 receptor in 293 cells: pharmacological and functional characterization.
Br. J. Pharmacol., 122 (2): 393-9. [PMID:9313952]
4. Hess JF, Derrick AW, MacNeil T, Borkowski JA. (1996)
The agonist selectivity of a mouse B1 bradykinin receptor differs from human and rabbit B1 receptors.
Immunopharmacology, 33 (1-3): 1-8. [PMID:8856107]
5. Jones C, Phillips E, Davis C, Arbuckle J, Yaqoob M, Burgess GM, Docherty RJ, Webb M, Bevan SJ, McIntyre P. (1999)
Molecular characterisation of cloned bradykinin B1 receptors from rat and human.
Eur J Pharmacol, 374: 423-433. [PMID:10422787]
6. MacNeil T, Feighner S, Hreniuk DL, Hess JF, Van der Ploeg LH. (1997)
Partial agonists and full antagonists at the human and murine bradykinin B1 receptors.
Can J Physiol Pharmacol, 75: 735-740. [PMID:9276157]
7. Menke JG, Borkowski JA, Bierilo KK, MacNeil T, Derrick AW, Schneck KA, Ransom RW, Strader CD, Linemeyer DL, Hess JF. (1994)
Expression cloning of a human B1 bradykinin receptor.
J Biol Chem, 269: 21583-21586. [PMID:8063797]