compound 5 [PMID: 29579323] [Ligand Id: 10038] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| TRPM4 in Human [GtoPdb: 496] [UniProtKB: Q8TD43] | ||||||||
| GtoPdb | In a patch clamp assay | - | 5.74 | pIC50 | 1800 | nM | IC50 | Br J Pharmacol (2018) 175: 2504-2519 [PMID:29579323] |
| GtoPdb | In a fluorescence cell‐based screening assay that monitors Na+ influx using the intracellular Na+ specific dye Asante natrium green‐II. | - | 5.82 | pIC50 | 1500 | nM | IC50 | Br J Pharmacol (2018) 175: 2504-2519 [PMID:29579323] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
