JAK inhibitor 20a [Ligand Id: 10147] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Janus kinase 1 in Human [GtoPdb: 2047] [UniProtKB: P23458] | ||||||||
| GtoPdb | - | - | 8.47 | pIC50 | 3.37 | nM | IC50 | J Med Chem (2018) 61: 10440-10462 [PMID:30460842] |
| Janus kinase 2 in Human [GtoPdb: 2048] [UniProtKB: O60674] | ||||||||
| GtoPdb | - | - | 7.53 | pIC50 | 29.6 | nM | IC50 | J Med Chem (2018) 61: 10440-10462 [PMID:30460842] |
| Janus kinase 3 in Human [GtoPdb: 2049] [UniProtKB: P52333] | ||||||||
| GtoPdb | - | - | 6.94 | pIC50 | 114.4 | nM | IC50 | J Med Chem (2018) 61: 10440-10462 [PMID:30460842] |
| tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597] | ||||||||
| GtoPdb | - | - | 7.13 | pIC50 | 73.7 | nM | IC50 | J Med Chem (2018) 61: 10440-10462 [PMID:30460842] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
