CpX [Ligand Id: 11313] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| LPA1 receptor in Human [GtoPdb: 272] [UniProtKB: Q92633] | ||||||||
| GtoPdb | - | - | 7.3 | pKi | 50 | nM | Ki | J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422] |
| GtoPdb | - | - | 7.5 | pEC50 | 31.6 | nM | EC50 | J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422] |
| LPA2 receptor in Human [GtoPdb: 273] [UniProtKB: Q9HBW0] | ||||||||
| GtoPdb | - | - | 7.1 | pKi | 79 | nM | Ki | J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422] |
| GtoPdb | - | - | 6.9 | pEC50 | 126 | nM | EC50 | J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422] |
| LPA3 receptor in Human [GtoPdb: 274] [UniProtKB: Q9UBY5] | ||||||||
| GtoPdb | - | - | 7.2 | pEC50 | 63 | nM | EC50 | J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
