XPC-5462 [Ligand Id: 13387] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Nav1.2 in Human [GtoPdb: 579] [UniProtKB: Q99250] | ||||||||
| GtoPdb | Concentration responses were measured at holding potentials where channels were maintained at fully inactivated potentials. | - | 7.96 | pIC50 | 10.9 | nM | IC50 | ACS Chem Neurosci (2024) 15: 1169-1184 [PMID:38359277] |
| Nav1.6 in Human [GtoPdb: 583] [UniProtKB: Q9UQD0] | ||||||||
| GtoPdb | Concentration responses were measured at holding potentials where channels were maintained at fully inactivated potentials. | - | 7.99 | pIC50 | 10.3 | nM | IC50 | ACS Chem Neurosci (2024) 15: 1169-1184 [PMID:38359277] |
| Nav1.6 in Mouse [GtoPdb: 583] [UniProtKB: Q9WTU3] | ||||||||
| GtoPdb | Concentration responses were measured at holding potentials where channels were maintained at fully inactivated potentials. | - | 7.86 | pIC50 | 13.7 | nM | IC50 | ACS Chem Neurosci (2024) 15: 1169-1184 [PMID:38359277] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
