MT-1207 [Ligand Id: 13442] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| 5-HT2A receptor in Human [GtoPdb: 6] [UniProtKB: P28223] | ||||||||
| GtoPdb | - | - | 10.1 | pKi | 0.08 | nM | Ki | J Med Chem (2024) 67: 16128-16144 [PMID:38968440] |
| GtoPdb | - | - | 9.54 | pIC50 | 0.29 | nM | IC50 | J Med Chem (2024) 67: 16128-16144 [PMID:38968440] |
| α1A-adrenoceptor in Human [GtoPdb: 22] [UniProtKB: P35348] | ||||||||
| GtoPdb | - | - | 10 | pIC50 | <0.1 | nM | IC50 | J Med Chem (2024) 67: 16128-16144 [PMID:38968440] |
| α1B-adrenoceptor in Human [GtoPdb: 23] [UniProtKB: P35368] | ||||||||
| GtoPdb | - | - | 10.07 | pKi | 0.09 | nM | Ki | J Med Chem (2024) 67: 16128-16144 [PMID:38968440] |
| GtoPdb | - | - | 9.82 | pIC50 | 0.15 | nM | IC50 | J Med Chem (2024) 67: 16128-16144 [PMID:38968440] |
| α1D-adrenoceptor in Human [GtoPdb: 24] [UniProtKB: P25100] | ||||||||
| GtoPdb | - | - | 9.16 | pKi | 0.69 | nM | Ki | J Med Chem (2024) 67: 16128-16144 [PMID:38968440] |
| GtoPdb | - | - | 8.85 | pIC50 | 1.4 | nM | IC50 | J Med Chem (2024) 67: 16128-16144 [PMID:38968440] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
