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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| carbonic anhydrase 1 in Human [GtoPdb: 2597] [UniProtKB: P00915] | ||||||||
| GtoPdb | - | - | 6.84 | pKi | 144.6 | nM | Ki | J Med Chem (2025) : [PMID:41150938] |
| histone deacetylase 3 in Human [GtoPdb: 2617] [UniProtKB: O15379] | ||||||||
| GtoPdb | - | - | 6.68 | pIC50 | 210 | nM | IC50 | J Med Chem (2025) : [PMID:41150938] |
| histone deacetylase 8 in Human [GtoPdb: 2619] [UniProtKB: Q9BY41] | ||||||||
| GtoPdb | - | - | 5.44 | pIC50 | 3600 | nM | IC50 | J Med Chem (2025) : [PMID:41150938] |
| carbonic anhydrase 12 in Human [GtoPdb: 2747] [UniProtKB: O43570] | ||||||||
| GtoPdb | - | - | 8.14 | pKi | 7.3 | nM | Ki | J Med Chem (2025) : [PMID:41150938] |
| carbonic anhydrase 9 in Human [GtoPdb: 3055] [UniProtKB: Q16790] | ||||||||
| GtoPdb | - | - | 7.51 | pKi | 31 | nM | Ki | J Med Chem (2025) : [PMID:41150938] |
| carbonic anhydrase 2 in Human [GtoPdb: 3092] [UniProtKB: P00918] | ||||||||
| GtoPdb | - | - | 8.13 | pKi | 7.4 | nM | Ki | J Med Chem (2025) : [PMID:41150938] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.