vexicitinib [Ligand Id: 14367] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Janus kinase 1 in Human [GtoPdb: 2047] [UniProtKB: P23458] | ||||||||
| GtoPdb | - | - | 7.7 | pIC50 | 20.04 | nM | IC50 | WO2022188796A1. Use of a compound containing a tricyclic heteroaryl group (2022) |
| Janus kinase 3 in Human [GtoPdb: 2049] [UniProtKB: P52333] | ||||||||
| GtoPdb | - | - | 8.84 | pIC50 | 1.43 | nM | IC50 | WO2022188796A1. Use of a compound containing a tricyclic heteroaryl group (2022) |
| tyrosine kinase 2 in Human [GtoPdb: 2269] [UniProtKB: P29597] | ||||||||
| GtoPdb | - | - | 9.09 | pIC50 | 0.82 | nM | IC50 | WO2022188796A1. Use of a compound containing a tricyclic heteroaryl group (2022) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
