BIM 23056 [Ligand Id: 2036] activity data from GtoPdb

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  • SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
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  • SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
  • SST3 receptor in Mouse [GtoPdb: 357] [UniProtKB: P30935]
  • SST3 receptor in Rat [GtoPdb: 357] [UniProtKB: P30936]
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  • SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
  • SST5 receptor in Mouse [GtoPdb: 359] [UniProtKB: O08858]
  • SST5 receptor in Rat [GtoPdb: 359] [UniProtKB: P30938]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
SST2 receptor in Human [GtoPdb: 356] [UniProtKB: P30874]
GtoPdb - - 6.7 pKi - - - Metab Clin Exp (1996) 45: 17-20 [PMID:8769372];
Naunyn Schmiedebergs Arch Pharmacol (1998) 357: 483-9 [PMID:9650799];
Naunyn Schmiedebergs Arch Pharmacol (1999) 360: 488-99 [PMID:10598788];
Eur J Pharmacol (1998) 348: 311-20 [PMID:9652348]
SST3 receptor in Human [GtoPdb: 357] [UniProtKB: P32745]
GtoPdb - - 7.2 pKi - - - Naunyn Schmiedebergs Arch Pharmacol (1998) 357: 483-9 [PMID:9650799];
Naunyn Schmiedebergs Arch Pharmacol (1999) 360: 488-99 [PMID:10598788]
SST3 receptor in Mouse [GtoPdb: 357] [UniProtKB: P30935]
GtoPdb - - 10.7 pIC50 - - - Mol Pharmacol (1993) 43: 838-44 [PMID:8100350]
SST3 receptor in Rat [GtoPdb: 357] [UniProtKB: P30936]
GtoPdb - - 6.5 pIC50 - - - J Neurochem (1997) 68: 2263-72 [PMID:9166718]
SST5 receptor in Human [GtoPdb: 359] [UniProtKB: P35346]
GtoPdb - - 8.3 pKi - - - Naunyn Schmiedebergs Arch Pharmacol (1998) 357: 483-9 [PMID:9650799];
Naunyn Schmiedebergs Arch Pharmacol (1999) 360: 488-99 [PMID:10598788];
Rev Physiol Biochem Pharmacol (1998) 133: 55-108 [PMID:9600011];
Endocrinology (1994) 135: 2814-7 [PMID:7988476];
Eur J Pharmacol (1998) 348: 311-20 [PMID:9652348]
GtoPdb - - 8.3 pKi - - Ki
SST5 receptor in Mouse [GtoPdb: 359] [UniProtKB: O08858]
GtoPdb - - 7.9 pKd - - - Neuropharmacology (2000) 39: 1451-62 [PMID:10818261]
SST5 receptor in Rat [GtoPdb: 359] [UniProtKB: P30938]
GtoPdb - - 6.3 pKi - - - Rev Physiol Biochem Pharmacol (1998) 133: 55-108 [PMID:9600011]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.