Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Kv1.1 in Rat [GtoPdb: 538] [UniProtKB: P10499] | ||||||||
| GtoPdb | - | - | 10.8 | pIC50 | - | - | - | Mol Pharmacol (1994) 45: 1227-34 [PMID:7517498] |
| Kv1.3 in Rat [GtoPdb: 540] [UniProtKB: P15384] | ||||||||
| GtoPdb | - | - | 12 | pIC50 | - | - | - |
J Biol Chem (1998) 273: 32697-707 [PMID:9830012]; Biochemistry (2003) 42: 13698-707 [PMID:14622016]; Int J Pept Protein Res (1995) 46: 354-8 [PMID:8567178] |
| Kv1.6 in Rat [GtoPdb: 543] [UniProtKB: P17659] | ||||||||
| GtoPdb | - | - | 9.8 | pIC50 | - | - | - | J Biol Chem (1998) 273: 32697-707 [PMID:9830012] |
| Kv1.7 in Mouse [GtoPdb: 544] [UniProtKB: Q17ST2] | ||||||||
| GtoPdb | - | - | 7.9 | pIC50 | - | - | - | J Biol Chem (1998) 273: 5851-7 [PMID:9488722] |
| Kv3.2 in Human [GtoPdb: 549] [UniProtKB: Q96PR1] | ||||||||
| GtoPdb | - | - | 9.5 | pIC50 | - | - | - | Mol Pharmacol (2005) 67: 1513-21 [PMID:15709110] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.