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1
_lig_chart_1
α1A-adrenoceptor
Rat
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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α1A-adrenoceptor in Rat [GtoPdb: 22] [UniProtKB: P43140] | ||||||||
GtoPdb | - | - | 5 | pKi | 10000 | nM | Ki | J. Biol. Chem. (2003) 278: 34451-7 [PMID:12824165] |
α1B-adrenoceptor in Human [GtoPdb: 23] [UniProtKB: P35368] | ||||||||
GtoPdb | - | - | 8.4 | pKi | - | - | - | J. Biol. Chem. (2004) 279: 35326-33 [PMID:15194691] |
α1B-adrenoceptor in Rat [GtoPdb: 23] [UniProtKB: P15823] | ||||||||
GtoPdb | - | - | 9.1 | pIC50 | 0.8 | nM | IC50 | Eur. J. Pharmacol. (2005) 508: 183-92 [PMID:15680270] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.