rho-TIA [Ligand Id: 507] activity data from GtoPdb

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  • α1A-adrenoceptor in Rat [GtoPdb: 22] [UniProtKB: P43140]
  • This target only has 1 pki data point
1 _lig_chart_1 α1A-adrenoceptor Rat
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  • α1B-adrenoceptor in Human [GtoPdb: 23] [UniProtKB: P35368]
  • α1B-adrenoceptor in Rat [GtoPdb: 23] [UniProtKB: P15823]
  • This target only has 1 pki data point
2 _lig_chart_2 α1B-adrenoceptor HumanRat
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
α1A-adrenoceptor in Rat [GtoPdb: 22] [UniProtKB: P43140]
GtoPdb - - 5 pKi 10000 nM Ki J. Biol. Chem. (2003) 278: 34451-7 [PMID:12824165]
α1B-adrenoceptor in Human [GtoPdb: 23] [UniProtKB: P35368]
GtoPdb - - 8.4 pKi - - - J. Biol. Chem. (2004) 279: 35326-33 [PMID:15194691]
α1B-adrenoceptor in Rat [GtoPdb: 23] [UniProtKB: P15823]
GtoPdb - - 9.1 pIC50 0.8 nM IC50 Eur. J. Pharmacol. (2005) 508: 183-92 [PMID:15680270]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.