galanin [Ligand Id: 6129] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211] | ||||||||
| GtoPdb | - | - | 9.1 | pKd | 0.8 | nM | Kd | Proc Natl Acad Sci USA (1994) 91: 9780-3 [PMID:7524088] |
| GtoPdb | - | - | 10.6 | pKi | 0.03 | nM | Ki |
J Pharmacol Exp Ther (1998) 287: 448-56 [PMID:9808667]; Peptides (1998) 19: 1771-81 [PMID:9880084]; Proc Natl Acad Sci USA (1994) 91: 9780-3 [PMID:7524088] |
| GtoPdb | - | - | 9.85 | pIC50 | 0.14 | nM | IC50 |
Biochem Biophys Res Commun (1997) 233: 823-8 [PMID:9168941]; Brain Res Mol Brain Res (1998) 58: 156-69 [PMID:9685625] |
| GAL1 receptor in Rat [GtoPdb: 243] [UniProtKB: Q62805] | ||||||||
| GtoPdb | - | - | 9.13 | pKd | 0.74 | nM | Kd | Regul Pept (1996) 62: 47-52 [PMID:8738882] |
| GtoPdb | - | - | 10 | pKi | 0.1 | nM | Ki |
J Biol Chem (1997) 272: 24612-6 [PMID:9305929]; J Biol Chem (1998) 273: 23321-6 [PMID:9722565]; Brain Res Mol Brain Res (1995) 34: 179-89 [PMID:8750821]; J Mol Neurosci (1995) 6: 33-41 [PMID:8562318] |
| GtoPdb | - | - | 10.22 | pIC50 | 0.06 | nM | IC50 |
Biochem Biophys Res Commun (1997) 233: 823-8 [PMID:9168941]; FEBS Lett (1997) 405: 285-90 [PMID:9108306] |
| GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603] | ||||||||
| GtoPdb | - | - | 9.02 | pKi | 0.95 | nM | Ki | Peptides (1998) 19: 1771-81 [PMID:9880084] |
| GtoPdb | - | - | 9.46 | pIC50 | 0.35 | nM | IC50 | Brain Res Mol Brain Res (1998) 58: 156-69 [PMID:9685625] |
| GtoPdb | - | - | 8.09 | pEC50 | 8.12 | nM | EC50 | Peptides (1998) 19: 1771-81 [PMID:9880084] |
| GAL2 receptor in Rat [GtoPdb: 244] [UniProtKB: O08726] | ||||||||
| GtoPdb | - | - | 9.3 | pKi | 0.5 | nM | Ki |
J Biol Chem (1997) 272: 24612-6 [PMID:9305929]; J Biol Chem (1998) 273: 23321-6 [PMID:9722565] |
| GtoPdb | - | - | 9.43 | pIC50 | 0.37 | nM | IC50 |
Brain Res Mol Brain Res (1997) 51: 49-59 [PMID:9427506]; FEBS Lett (1997) 405: 285-90 [PMID:9108306] |
| GtoPdb | - | - | 7.74 | pEC50 | 18 | nM | EC50 | J Biol Chem (1997) 272: 24612-6 [PMID:9305929] |
| GAL3 receptor in Human [GtoPdb: 245] [UniProtKB: O60755] | ||||||||
| GtoPdb | - | - | 8.01 | pKi | 9.77 | nM | Ki |
J Biol Chem (1998) 273: 23321-6 [PMID:9722565]; Peptides (1998) 19: 1771-81 [PMID:9880084] |
| GtoPdb | - | - | 7.92 | pIC50 | 12 | nM | IC50 | J Neurochem (1998) 71: 2239-51 [PMID:9832121] |
| GAL3 receptor in Rat [GtoPdb: 245] [UniProtKB: O88626] | ||||||||
| GtoPdb | - | - | 8.14 | pKi | 7.24 | nM | Ki | J Biol Chem (1998) 273: 23321-6 [PMID:9722565] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
