seltorexant [Ligand Id: 9308] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| OX1 receptor in Human [GtoPdb: 321] [UniProtKB: O43613] | ||||||||
| GtoPdb | In vitro radioligand binding assay | - | 6.1 | pKi | 794 | nM | Ki | J Pharmacol Exp Ther (2015) 354: 471-82 [PMID:26177655] |
| OX1 receptor in Rat [GtoPdb: 321] [UniProtKB: P56718] | ||||||||
| GtoPdb | In vitro radioligand binding assay | - | 6.2 | pKi | 630 | nM | Ki | J Pharmacol Exp Ther (2015) 354: 471-82 [PMID:26177655] |
| OX2 receptor in Human [GtoPdb: 322] [UniProtKB: O43614] | ||||||||
| GtoPdb | In vitro radioligand binding assay | - | 8 | pKi | 10 | nM | Ki | J Pharmacol Exp Ther (2015) 354: 471-82 [PMID:26177655] |
| OX2 receptor in Rat [GtoPdb: 322] [UniProtKB: P56719] | ||||||||
| GtoPdb | In vitro radioligand binding assay | - | 8.1 | pKi | 7.9 | nM | Ki | J Pharmacol Exp Ther (2015) 354: 471-82 [PMID:26177655] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
