surufatinib [Ligand Id: 9769] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362]
There should be some charts here, you may need to enable JavaScript!
  • kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
fibroblast growth factor receptor 1 in Human [GtoPdb: 1808] [UniProtKB: P11362]
GtoPdb Using a Transcreener FP technology assay. - 7.28 pIC50 53 nM IC50 WO2011060746. Compound, certain novel forms thereof, pharmaceutical compositions thereof and methods for preparation and use (2011)
kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968]
GtoPdb In a biochemical assay using recombinant KDR kinase catalytic domain. - 7.68 pIC50 21 nM IC50 WO2011060746. Compound, certain novel forms thereof, pharmaceutical compositions thereof and methods for preparation and use (2011)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.