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Synonyms: [125I]-Hpp-desArg9HOE140
Compound class:
Peptide
Comment: Radiolabelled analogue of icatibant (HOE 140), a synthetic analogue of bradykinin.
Ligand Activity Visualisation ChartsThese are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts. ✖ |
| References |
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1. de Sousa Buck H, Ongali B, Thibault G, Lindsey CJ, Couture R. (2002)
Autoradiographic detection of kinin receptors in the human medulla of control, hypertensive, and diabetic donors. Can J Physiol Pharmacol, 80 (4): 249-57. [PMID:12025957] |
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2. Ongali B, Hellal F, Rodi D, Plotkine M, Marchand-Verrecchia C, Pruneau D, Couture R. (2006)
Autoradiographic analysis of mouse brain kinin B1 and B2 receptors after closed head trauma and ability of Anatibant mesylate to cross the blood-brain barrier. J Neurotrauma, 23 (5): 696-707. [PMID:16689671] |
