INSL5 analogue 13   Click here for help

GtoPdb Ligand ID: 11915

Compound class: Peptide
Comment: This is an INSL5 analogue that has a simplified A-chain connected to the B-chain by two disulfide bonds [1]. Its A-chain peptide sequence is hINSL5: A8-21 (T15K).
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
RXFP4 Hs Agonist Agonist 7.5 pKi - 2
pKi 7.5 [2]
RXFP4 Hs Agonist Agonist 7.7 pIC50 - 2
pIC50 7.7 [2]