MT-II

Ligand id: 1323

Name: MT-II

Structure and Physico-chemical Properties

2D Structure

View interactive charts of activity data from GtoPdb and ChEMBL (where available) across species

Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
MC4 receptor Hs Agonist Full agonist 8.2 – 8.8 pKi - 1-2,4
pKi 8.2 – 8.8 [1-2,4]
MC3 receptor Hs Agonist Full agonist 8.3 pKi - 1
pKi 8.3 [1]
MC1 receptor Hs Agonist Full agonist 9.4 pIC50 - 2-3
pIC50 9.4 [2-3]
MC5 receptor Hs Agonist Full agonist 9.0 pIC50 - 3
pIC50 9.0 [3]