neurotensin

Ligand id: 1579

Name: neurotensin

Species: Human, Mouse, Rat, Bovine

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Structure and Physico-chemical Properties

2D Structure
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Natural/Endogenous Targets
Target
NTS1 receptor
NTS2 receptor
Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
NTS1 receptor Rn Agonist Full agonist 8.2 – 10.0 pKi - 3,5,8
pKi 8.2 – 10.0 [3,5,8]
NTS1 receptor Hs Agonist Full agonist 8.3 – 9.7 pKi - 3,7
pKi 8.3 – 9.7 [3,7]
NTS2 receptor Hs Agonist Full agonist 8.8 pKi - 7
pKi 8.8 [7]
NTS2 receptor Mm Agonist Full agonist 8.5 – 8.7 pIC50 - 1
pIC50 8.5 – 8.7 [1]
NTS2 receptor Rn Agonist Full agonist 8.2 pIC50 - 2
pIC50 8.2 [2]
Additional information and targets (data relate to human unless otherwise stated)
Description Data Reference
Ligand mentioned in the following text fields