VPAC2 receptor
|
|
|
Hs |
Agonist |
Partial agonist |
8.3 – 8.4 |
pEC50 |
- |
1 |
|
⤷ |
pEC50
8.4
(EC50 4.4x10-9 M)
[1]
Description: inhibition of calcium influx stimulated by 30nM VIP in CHO cells stably expressing recombinant receptor
pEC50
8.3
(EC50 4.9x10-9 M)
[1]
Description: cyclic AMP formation in CHO cells stably expressing recombinant receptor
|
PAC1 receptor
|
|
|
Hs |
Agonist |
Agonist |
7.1 |
pEC50 |
- |
1 |
|
⤷ |
pEC50
7.1
(EC50 7.13x10-8 M)
[1]
Description: cyclic AMP formation in CHO cells stably expressing recombinant receptor
|
VPAC1 receptor
|
|
|
Hs |
Agonist |
Agonist |
<5.5 – 8.1 |
pEC50 |
- |
1 |
|
⤷ |
pEC50
8.1
(EC50 8.04x10-9 M)
[1]
Description: cyclic AMP formation in CHO cells stably expressing recombinant receptor
pEC50
<5.5
(EC50 >3x10-6 M)
[1]
Description: calcium influx in CHO cells stably expressing recombinant receptor
|
VPAC2 receptor
|
|
|
Hs |
Antagonist |
Antagonist |
8.7 |
pIC50 |
- |
2 |
|
⤷ |
pIC50
8.7
(IC50 2x10-9 M)
[2]
Description: inhibition of [125I]Ro25 1553 binding to membranes from CHO cells stably expressing the recombinant receptor
|
VPAC2 receptor
|
|
|
Hs |
Agonist |
Partial agonist |
7.6 |
pIC50 |
- |
1 |
|
⤷ |
pIC50
7.6
(IC50 2.29x10-8 M)
[1]
Description: inhibition of cyclic AMP formation stimulated by 0.3nM VIP in CHO cells stably expressing recombinant receptor
|
VPAC1 receptor
|
|
|
Hs |
Agonist |
Partial agonist |
6.7 |
pIC50 |
- |
2 |
|
⤷ |
pIC50
6.7
(IC50 2x10-7 M)
[2]
Description: inhibition of [125I]-VIP binding to membranes from CHO cells stably expressing the recombinant receptor
|