[Ala1,3,11,15]ET-1   Click here for help

GtoPdb Ligand ID: 3837

Synonyms: [Ala1,3,11,15]endothelin-1
Comment: Synthetic analogue of ET-1
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
ETB receptor Hs Agonist Full agonist 8.7 – 9.2 pKd - 1
pKd 8.7 – 9.2 (Kd 1.82x10-9 – 6.43x10-10 M) [1]