nicotinic acetylcholine receptor α7 subunit
|
|
|
Hs |
Agonist |
Full agonist |
12.2 |
pKd |
- |
|
|
⤷ |
pKd
12.2
(Kd 6x10-13 M)
(α7)5
|
nicotinic acetylcholine receptor α2 subunit
|
|
|
Rn |
Agonist |
Full agonist |
10.1 – 11.0 |
pKd |
- |
|
|
⤷ |
pKd
10.7 – 11.0
(Kd 2.1x10-11 – 1x10-11 M)
α2β2
pKd
10.1 – 10.1
(Kd 8.7x10-11 – 8.4x10-11 M)
α2β4
|
nicotinic acetylcholine receptor α6 subunit
|
|
|
Ggal |
Agonist |
Full agonist |
10.5 |
pKd |
- |
|
|
⤷ |
pKd
10.5
(Kd 3.5x10-11 M)
native α6β4*
|
nicotinic acetylcholine receptor α3 subunit
|
|
|
Hs |
Agonist |
Full agonist |
9.6 – 11.1 |
pKd |
- |
|
|
⤷ |
pKd
11.1
(Kd 7x10-12 M)
α3β2
pKd
9.6
(Kd 2.3x10-10 M)
α3β4
|
nicotinic acetylcholine receptor α2 subunit
|
|
|
Hs |
Agonist |
Full agonist |
10.4 |
pKd |
- |
|
|
⤷ |
pKd
10.4
(Kd 4.2x10-11 M)
α2β4
|
nicotinic acetylcholine receptor α4 subunit
|
|
|
Hs |
Agonist |
Full agonist |
9.7 – 11.0 |
pKd |
- |
|
|
⤷ |
pKd
10.5 – 11.0
(Kd 3.3x10-11 – 1x10-11 M)
α4β2
pKd
9.7
(Kd 1.87x10-10 M)
α4β4
|
nicotinic acetylcholine receptor α3 subunit
|
|
|
Rn |
Agonist |
Full agonist |
9.5 – 10.9 |
pKd |
- |
|
|
⤷ |
pKd
10.5 – 10.9
(Kd 3.4x10-11 – 1.4x10-11 M)
α3β2
pKd
9.5 – 9.5
(Kd 3.04x10-10 – 2.9x10-10 M)
α3β4
|
nicotinic acetylcholine receptor α8 subunit (avian)
|
|
|
Hs |
None |
- |
9.7 |
pKd |
- |
|
|
⤷ |
pKd
9.7
(Kd 2x10-10 M)
(α8)5
|
nicotinic acetylcholine receptor α4 subunit
|
|
|
Rn |
Agonist |
Full agonist |
9.0 – 9.5 |
pKd |
- |
|
|
⤷ |
pKd
9.3 – 9.5
(Kd 4.6x10-10 – 3x10-10 M)
α4β2
pKd
9.0 – 9.1
(Kd 9.4x10-10 – 8.5x10-10 M)
α4β4
|