Tyr3-octreotide   Click here for help

GtoPdb Ligand ID: 5649

Synonyms: SMS 204,090 | TOC | Tyr3-SMS 201,995
Comment: This is an analogue of octreotide. Tyr3-octreotide can be radio-labelled (e.g. with technetium-99) for use in nuclear medicine to image neuroendocrine tumours expressing the somatostatin receptor [1].
Bioactivity Comments
Although we have been unable to find peer reviewed affinity data for the interaction of this analogue with any of the the somatostatin receptors, we have tagged somatostatin receptor 2 as primary molecular target for data retrieval puproses only.
Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
SST2 receptor Primary target of this compound Hs Agonist Agonist - - -