View interactive charts of activity data from GtoPdb and ChEMBL (where available) across species

Selectivity at GPCRs
Key to terms and symbols		Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference BB1 receptor Hs Antagonist Antagonist 6.2 – 6.3 pIC50 - 1 ⤷ pIC50 6.2 – 6.3 (IC50 6.3x10-7 – 4.68x10-7 M) [1] BB2 receptor Hs Antagonist Antagonist 5.0 – 5.5 pIC50 - 1 ⤷ pIC50 5.0 – 5.5 (IC50 1x10-5 – 3.47x10-6 M) [1]