Ac-Phe-Trp-Ala-His(τBZL)-Nip-Gly-Arg-NH2   Click here for help

GtoPdb Ligand ID: 6191

Comment: This is a mix of stereoisomers; see discussion on analogue 34 in [1].
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
BB3 receptor Hs Agonist Full agonist 6.4 – 8.2 pEC50 - 1-3
pEC50 6.4 – 8.2 (EC50 3.98x10-7 – 6.9x10-9 M) [1-3]
BB3 receptor Hs Agonist Full agonist 6.2 – 7.3 pIC50 - 2-3
pIC50 6.2 – 7.3 (IC50 5.72x10-7 – 4.9x10-8 M) [2-3]