Ac-Phe-Trp-Ala-His(τBZL)-Nip-Gly-Arg-NH2   Click here for help

GtoPdb Ligand ID: 6191

Comment: This is a mix of stereoisomers; see discussion on analogue 34 in [1].
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1. Boyle RG, Humphries J, Mitchell T, Showell GA, Apaya R, Iijima H, Shimada H, Arai T, Ueno H, Usui Y et al.. (2005)
The design of a new potent and selective ligand for the orphan bombesin receptor subtype 3 (BRS3).
J Pept Sci, 11 (3): 136-41. [PMID:15635635]
2. Gonzalez N, Hocart SJ, Portal-Nuñez S, Mantey SA, Nakagawa T, Zudaire E, Coy DH, Jensen RT. (2008)
Molecular basis for agonist selectivity and activation of the orphan bombesin receptor subtype 3 receptor.
J Pharmacol Exp Ther, 324 (2): 463-74. [PMID:18006692]
3. Sancho V, Moody TW, Mantey SA, Di Florio A, Uehara H, Coy DH, Jensen RT. (2010)
Pharmacology of putative selective hBRS-3 receptor agonists for human bombesin receptors (BnR): affinities, potencies and selectivity in multiple native and BnR transfected cells.
Peptides, 31 (8): 1569-78. [PMID:20438784]