[Leu9,des-Arg10]kallidin   Click here for help

GtoPdb Ligand ID: 642

Synonyms: [Lys,Leu8,des-Arg9]bradykinin | Lys-[Leu8][des-Arg9]BK | Lys-[Leu8][des-Arg9]bradykinin
Click here for help
Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
B1 receptor Mm Antagonist Antagonist 7.0 pA2 - 1
pA2 7.0 [1]
B1 receptor Hs Antagonist Antagonist 9.1 – 9.3 pKi - 2-3
pKi 9.1 – 9.3 [2-3]
B1 receptor Mm Antagonist Antagonist 8.1 pKi - 4
pKi 8.1 [4]
B1 receptor Hs Antagonist Antagonist 8.9 pIC50 - 5
pIC50 8.9 [5]