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Synonyms: [Lys,Leu8,des-Arg9]bradykinin | Lys-[Leu8][des-Arg9]BK | Lys-[Leu8][des-Arg9]bradykinin
Compound class:
Peptide or derivative
Ligand Activity Visualisation ChartsThese are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts. ✖ |
| References |
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1. Allogho SN, Gobeil F, Pheng LH, Nguyen-Le XK, Neugebauer W, Regoli D. (1995)
Kinin B1 and B2 receptors in the mouse. Can J Physiol Pharmacol, 73 (12): 1759-64. [PMID:8834490] |
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2. Austin CE, Faussner A, Robinson HE, Chakravarty S, Kyle DJ, Bathon JM, Proud D. (1997)
Stable expression of the human kinin B1 receptor in Chinese hamster ovary cells. Characterization of ligand binding and effector pathways. J Biol Chem, 272 (17): 11420-5. [PMID:9111052] |
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3. Bastian S, Loillier B, Paquet JL, Pruneau D. (1997)
Stable expression of human kinin B1 receptor in 293 cells: pharmacological and functional characterization. Br J Pharmacol, 122 (2): 393-9. [PMID:9313952] |
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4. Hess JF, Derrick AW, MacNeil T, Borkowski JA. (1996)
The agonist selectivity of a mouse B1 bradykinin receptor differs from human and rabbit B1 receptors. Immunopharmacology, 33 (1-3): 1-8. [PMID:8856107] |
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5. Menke JG, Borkowski JA, Bierilo KK, MacNeil T, Derrick AW, Schneck KA, Ransom RW, Strader CD, Linemeyer DL, Hess JF. (1994)
Expression cloning of a human B1 bradykinin receptor. J Biol Chem, 269: 21583-21586. [PMID:8063797] |
